NanoBRET™ TE Intracellular Kinase Cell-Based Assay Services Target List
Targets in blue letters have been successfully validated at Carna.
For targets in grey letters, please contact us for its turnaround time.
For targets in grey letters, please contact us for its turnaround time.
Kinase Name | Data Sample | Kinase Name | Data Sample |
---|---|---|---|
AAK1 |
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LCK |
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ABL1(ABL) |
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LIMK1 |
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ABL1(ABL)[E255K] | LIMK2 |
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ABL1(ABL)[F317I] | LRRK2 |
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ABL1(ABL)[F317L] | LRRK2[G2019S] | ||
ABL1(ABL)[H396P] | LRRK2[I2020T] | ||
ABL1(ABL)[M351T] | LRRK2[R1441C] | ||
ABL1(ABL)[Q252H] | LTK |
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ABL1(ABL)[T315I] | LYN |
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ABL1(ABL)[Y253F] | MAP2K6 | ||
ABL2(ARG) | MAP3K10(MLK2) |
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ACVR1(ALK2) |
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MAP3K11(MLK3) |
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ACVR1(ALK2)[G328V] | MAP3K12(DLK) |
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ACVR1(ALK2)[G356D] | MAP3K13(LZK) | ||
ACVR1(ALK2)[Q207D] | MAP3K19 |
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ACVR1(ALK2)[R206H] | MAP3K2 | ||
ACVRL1(ALK1) |
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MAP3K21(MLK4) | |
ADK | MAP3K3 | ||
AKT1 | MAP3K4 |
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AKT1 [E17K] | MAP3K9(MLK1) |
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AKT2 |
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MAP4K1(HPK1) |
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AKT2[E17K] | MAP4K2 |
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AKT3[E17K] | MAP4K3 |
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AKT3[G171R] | MAP4K5 |
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ALK |
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MAPK11(p38β) |
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ALK4(ACVR1B) |
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MAPK14 (p38α)[T106M] | |
AurA |
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MAPK14(p38α) |
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AurB |
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MAPK4 |
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AurC |
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MAPK6 |
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AXL |
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MARK2 |
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BLK |
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MARK3 | |
BMP2K |
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MARK4 |
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BMPR1A | MAST3 | ||
BMX |
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MAST4 | |
BRAF[V600E] | MELK |
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BRK (PTK6) |
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MELK [T460M] | |
BRSK1 | MER (MERTK) |
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BRSK2 |
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MER(MERTK)[A708S] | |
BTK |
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MET |
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BTK E41K] | MET[D1228H] | ||
BTK P190K] | MET[D1228N] | ||
BTK[C481S] |
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MET[F1200I] | |
CAMK1 | MET[M1250T] | ||
CAMK1D |
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MET[P991S] | |
CAMK1G | MET[T1173I] | ||
CAMK2A(CaMK2α) | MET[T992I] | ||
CAMK2D(CaMK2δ) | MET[V1092I] | ||
CAMK2G(CaMK2γ) | MET[Y1230A] | ||
CDK10/CycL2 | MET[Y1230C] | ||
CDK11A/Cyc K | MET[Y1230D] | ||
CDK11A/Cyc L2 | MET[Y1230H] | ||
CDK14/Cyc Y |
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MET[Y1235D] | |
CDK15/Cyc Y | MKNK2(MNK2) | ||
CDK16(PCTAIRE1)/CycY |
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MLTK (ZAK) | |
CDK17/Cyc Y |
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MOK | |
CDK18/Cyc Y |
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MUSK |
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CDK19/Cyc C | MYLK2(skMLCK) |
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CDK1/CycB1 (CDC2/CycB1) |
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MYLK3 | |
CDK1/CycE1 (CDC2/CycE1) | MYLK4 |
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CDK20/Cyc H | NEK1 | ||
CDK2/CycA1 |
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NEK11 | |
CDK2/CycE1 |
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NEK2 |
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CDK3/Cyc E1 |
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NEK3 |
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CDK4/Cyc D1 |
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NEK4 | |
CDK4/Cyc D3 |
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NEK5 | |
CDK5 |
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NEK6 | |
CDK5/CDK5R1 |
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NEK9 |
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CDK5/CDK5R2 | NIM1K(MGC42105) | ||
CDK6/CycD1 |
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NLK | |
CDK6/CycD3 |
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NRK | |
CDK7 |
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NuaK1 (ARK5) |
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CDK7/Cyc H |
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NuaK2 | |
CDK8/Cyc C |
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PAK4 |
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CDK9/CycK |
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PAK6 | |
CDK9/CycT1 |
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PAK7(PAK5) |
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CDKL1 | PDGFRA[V561D] |
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CDKL2 | PHKG1 |
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CDKL3 | PHKG2 | ||
CDKL5 | PIK3C3 | ||
CHEK1(CHK1) |
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PIK3CA [M1043I]/PIK3R1 | |
CHEK2(CHK2) | PIK3CA[C420R]/PIK3R1 | ||
CLK1 |
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PIK3CA[E542K]/PIK3R1 | |
CLK2 |
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PIK3CA[E545A]/PIK3R1 | |
CLK4 |
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PIK3CA[E545K]/PIK3R1 |
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COQ8B | PIK3CA[H1047L]/PIK3R1 |
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CSF1R(FMS) |
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PIK3CA[H1047R]/PIK3R1 |
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CSK |
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PIK3CA[H1047Y]/PIK3R1 | |
CSNK1A1L | PIK3CA[I800L]/PIK3R1 | ||
CSNK1D(CK1δ) |
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PIK3CA[Q546K]/PIK3R1 | |
CSNK1E(CK1ε) | PIK3CA/PIK3R1 |
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CSNK1G2(CK1γ2) |
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PIK3CB/PIK3R1 | |
CSNK2A1 |
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PIK3CD/PIK3R1 | |
CSNK2A2 |
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PIKFYVE(PIP5K3) |
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DAPK2 | PIM3 | ||
DCLK3 | PIP4K2C |
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DDR1 |
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PIP5K1B | |
DDR2 |
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PKACα(PRKACA) |
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DDR2[N456S] | PKACβ (PRKACB) | ||
DMPK(DMPK1) | PKMYT1(MYT1) |
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DYRK1A |
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PLK2 | |
DYRK1B |
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PLK3 | |
DYRK2 | PLK4 |
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EIF2AK4(GCN2) _Domain2 | PRKAA1 | ||
EPHA1 |
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PRKAA2 |
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EPHA2 |
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PRKCE(PKCε) | |
EPHA3 | PRKG2(CGK2) | ||
EPHA4 |
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PRKX |
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EPHA5 |
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PYK2 (PTK2B) |
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EPHA6 |
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RET |
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EPHA7 |
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RET[M918T] | |
EPHA8 |
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RET[V804L] | |
EPHB1 | RET[V804M] | ||
EPHB2 |
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RIOK2 |
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EPHB3 |
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RIPK1 |
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EPHB4 |
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RIPK2 |
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Erk1 (MAPK3) |
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RON |
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Erk2(MAPK1) |
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RPS6KA4(MSK2) |
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ERN1 |
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RSK1 (RPS6KA1) |
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ERN2 | RSK2(RPS6KA3) |
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FAK (PTK2) |
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RSK2(RPS6KA3)[I416V] | |
FER |
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RSK2(RPS6KA3)[L608F] | |
FES | RSK3 (RPS6KA2) |
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FGFR1 |
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RSK4 (RPS6KA6) |
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FGFR2 |
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SBK3 | |
FGFR2[K659M] |
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SGK1 | |
FGFR2[L617F] |
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SGK2 | |
FGFR2[L617V] |
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SIK1 |
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FGFR2[M537I] |
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SIK2 (QIK, SNF1LK2) |
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FGFR2[N549H] |
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SIK3(QSK) |
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FGFR2[N549K] |
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SLK |
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FGFR2[V564F] |
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SNRK | |
FGFR3 |
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SRC |
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FGFR3[G697C] |
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SRMS(SRM) | |
FGFR3[V555M] |
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STK10(LOK) |
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FGFR4 |
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STK11 |
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FGR |
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STK16 |
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FLT1 |
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STK17B | |
FLT3 |
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STK24(MST3) | |
FLT3[D835H] | STK26(MST4) | ||
FLT3[D835V] | STK3(MST2) | ||
FLT3[D835Y] | STK32A | ||
FLT3[K663Q] | STK32B |
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FLT3[N841I] | STK33 |
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FLT3[R834Q] | STK35 |
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FRK |
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STK36 | |
FYN |
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STK38(NDR1) |
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FYN[Y531F] | STK38L(NDR2) | ||
GAK |
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STK4(MST1) |
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GSK3A(GSK3α) |
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TBK1 |
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GSK3B(GSK3β) |
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TEC |
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HCK | TEK(TIE2) |
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HIPK2 | TEK(TIE2)[A1124V] | ||
HIPK3 | TEK(TIE2)[P883A] | ||
HIPK4 | TEK(TIE2)[R849W] | ||
ICK | TEK(TIE2)[Y1108F] | ||
IGF1R |
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TEK(TIE2)[Y897C] | |
IKBKE(IKKε) |
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TEK(TIE2)[Y897S] | |
INSR |
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TESK1 |
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IRAK1 | TGFBR2 | ||
IRAK3 |
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TIE1 |
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IRAK4 |
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TLK1 | |
ITK |
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TLK2 | |
JAK1 |
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TNK1 |
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JAK1_JH1 Domain |
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TNK2 (ACK) |
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JAK2 |
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TNNI3K(HH498) | |
JAK2[V617F] |
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TRKA (NTRK1) |
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JAK2_JH1 Domain |
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TRKA(NTRK1)[G667C] | |
JAK3 |
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TRKB(NTRK2) |
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JNK1(MAPK8) |
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TSSK1B | |
JNK2(MAPK9) |
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TTK |
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JNK3 |
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TXK |
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KIT |
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TYK2 |
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KIT[A829P] | TYK2_JH1 Domain |
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KIT[D816H] | TYK2_JH2 Domain |
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KIT[D816V] |
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TYRO3 |
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KIT[L576P] | ULK1 |
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KIT[V559D,T670I] | ULK2 |
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KIT[V559D,V654A] | ULK3 |
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KIT[V559D] | WEE1 |
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LATS1 |
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WEE2 | |
LATS2 |
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YES1(YES) |
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