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- NanoBRET™ TE Intracellular Kinase Assay Services Target List
NanoBRET™ TE Intracellular Kinase Assay Services Target List
Target list for NanoBRET™ TE Intracellular Kinase Assay Services is shown below. Targets in blue text have been successfully validated at Carna and the study results will be delivered approximately in two weeks for IC50 determinations and approximately in three weeks for Residence Time Analysis. Please inquire regarding targets shown in grey text, as the turnaround time will vary.
Kinase Name
Data Sample
Kinase Name
Data Sample
Kinase Name
Data Sample
ABL1(ABL)[E255K]
ABL1(ABL)[F317I]
ABL1(ABL)[F317L]
ABL1(ABL)[H396P]
ABL1(ABL)[M351T]
ABL1(ABL)[Q252H]
ABL1(ABL)[T315I]
ABL1(ABL)[Y253F]
ACVR1(ALK2)[G328V]
ACVR1(ALK2)[G356D]
ACVR1(ALK2)[Q207D]
ACVR1(ALK2)[R206H]
ADK
AKT1[E17K]
AKT2[E17K]
AKT3[E17K]
AKT3[G171R]
BMPR1A
BTK[E41K]
BTK[P190K]
CAMK1G
(CaMK1γ)
CAMK2G(CaMK2γ)
CDK11A／CycK
CDK11A／CycL2
CDK19／CycC
CDK1／CycE1(CDC2/CycE1)
CDK5／CDK5R2
CSNK1E(CK1ε)
DDR2[N456S]
DMPK(DMPK1)
DYRK2
EIF2AK4(GCN2)_Domain2
EPHA3
FLT3[D835H]
FLT3[D835V]
FLT3[D835Y]
FLT3[K663Q]
FLT3[N841I]
FLT3[R834Q]
FYN[Y531F]
HCK
IRAK1
KIT[A829P]
KIT[D816H]
KIT[L576P]
KIT[V559D,T670I]
KIT[V559D,V654A]
KIT[V559D]
LRRK2[G2019S]
LRRK2[I2020T]
LRRK2[R1441C]
MAP2K6
MAP3K13(LZK)
MAPK14(p38α)[T106M]
MARK3
MELK[T460M]
MER(MERTK)[A708S]
MET[D1228H]
MET[D1228N]
MET[F1200I]
MET[M1250T]
MET[P991S]
MET[T1173I]
MET[T992I]
MET[V1092I]
MET[Y1230A]
MET[Y1230C]
MET[Y1230D]
MET[Y1230H]
MET[Y1235D]
MOK
NEK6
NRK
NuaK2
PIK3C3
PIK3CA[C420R]／PIK3R1
PIK3CA[E542K]／PIK3R1
PIK3CA[E545A]／PIK3R1
PIK3CA[H1047Y]／PIK3R1
PIK3CA[I800L]／PIK3R1
PIK3CA[M1043I]／PIK3R1
PIK3CA[Q546K]／PIK3R1
PIK3CB／PIK3R1
PIK3CD／PIK3R1
PIP5K1B
PKCβ1(PRKCB1)
PKCγ(PRKCG)
PKCη
(PRKCH)
PRKG2(CGK2)
RET[M918T]
RET[V804L]
RET[V804M]
RSK2(RPS6KA3)[I416V]
RSK2(RPS6KA3)[L608F]
SGK2
STK24(MST3)
STK26(MST4)
STK32A
TEK(TIE2)[A1124V]
TEK(TIE2)[P883A]
TEK(TIE2)[R849W]
TEK(TIE2)[Y1108F]
TEK(TIE2)[Y897C]
TEK(TIE2)[Y897S]
TGFBR2
TRKA(NTRK1)[G667C]
TSSK1B