| 2021年6月 | ||||||
| 日 | 月 | 火 | 水 | 木 | 金 | 土 |
|---|---|---|---|---|---|---|
| 1 | 2 | 3 | 4 | 5 | ||
| 6 | 7 | 8 | 9 | 10 | 11 | 12 |
| 13 | 14 | 15 | 16 | 17 | 18 | 19 |
| 20 | 21 | 22 | 23 | 24 | 25 | 26 |
| 27 | 28 | 29 | 30 | |||
| 2021年7月 | ||||||
| 日 | 月 | 火 | 水 | 木 | 金 | 土 |
|---|---|---|---|---|---|---|
| 1 | 2 | 3 | ||||
| 4 | 5 | 6 | 7 | 8 | 9 | 10 |
| 11 | 12 | 13 | 14 | 15 | 16 | 17 |
| 18 | 19 | 20 | 21 | 22 | 23 | 24 |
| 25 | 26 | 27 | 28 | 29 | 30 | 31 |
| 被験物質 受付締切日 | |
| MSA / IMAPTMアッセイ開始日 | |
| ELISA, ADP-Glo™, MSA(Preincubation)アッセイ開始日 |
以下のキナーゼをMobility Shift Assay、またはIMAP™で測定します。ATP濃度はKm値付近、または1mMで設定しています。化合物受領後、最短2週間で結果報告いたします。サービスのお申込は申込書にご記入の上、メールにてご提示下さい。
また、当社ではSlow Binderの評価に最適なPreincubation試験サービスも行なっています。詳しくはこちらをご覧下さい。
| 対象キナーゼ | グループ | 可能な測定メニュー(測定系: Mobility Shift Assay, IMAP™) |
使用キナーゼ (当社製品) |
|||||||
| セレクトパネル | ||||||||||
| ABL(ABL1) | TK | Km bin. | 1mM | Preincubation | TK | 08-001 | ||||
| ABL(ABL1)[E255K] | TK | Km bin. | 1mM | Preincubation | 08-094 | |||||
| ABL(ABL1)[T315I] | TK | Km bin. | 1mM | Preincubation | 08-093 | |||||
| ACK(TNK2) | TK | Km bin. | 1mM | 08-196 | ||||||
| AKT1 | STK | Km bin. | 1mM | Preincubation | STK | 01-101 | ||||
| AKT2 | STK | Km bin. | Preincubation | 01-102 | ||||||
| AKT3 | STK | Km bin. | Preincubation | 01-103 | ||||||
| ALK | TK | Km bin. | 1mM | Preincubation | 08-518 | |||||
| ALK[C1156Y] | TK | Km bin. | 1mM | Preincubation | 08-530 | |||||
| ALK[F1174L] | TK | Km bin. | 1mM | Preincubation | 08-519 | |||||
| ALK[G1202R] | TK | Km bin. | 1mM | Preincubation | 08-544 | |||||
| ALK[G1269A] | TK | Km bin. | 1mM | Preincubation | 08-537 | |||||
| ALK[L1196M] | TK | Km bin. | 1mM | Preincubation | 08-529 | |||||
| ALK[R1275Q] | TK | Km bin. | 1mM | Preincubation | 08-520 | |||||
| ALK[T1151_L1152insT] | TK | Km bin. | 1mM | 08-539 | ||||||
| AMPKα1/β1/γ1 (PRKAA1/B1/G1) | STK | Km bin. | 1mM | Preincubation | STK | 02-113 | ||||
| AMPKα2/β1/γ1 (PRKAA2/B1/G1) | STK | Km bin. | Preincubation | 02-114 | ||||||
| ARG(ABL2) | TK | Km bin. | 1mM | Preincubation | 08-102 | |||||
| AurA (AURKA) | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 05-101 | |||
| AurA(AURKA)/TPX2 | STK | Km bin. | Preincubation | 05-186 | ||||||
| AurB(AURKB)/INCENP | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 05-102 | ||||
| AurC (AURKC) | STK | Km bin. | 1mM | Cell Cycle | 05-103 | |||||
| AXL | TK | Km bin. | 1mM | 08-107 | ||||||
| BLK | TK | Km bin. | 1mM | 08-164 | ||||||
| BMX | TK | Km bin. | 1mM | Preincubation | 08-179 | |||||
| BRAF | STK |
1mM (Cascade) |
MAPK (Cascade) |
09-122 | ||||||
| BRAF[V600E] | STK |
1mM (Cascade) |
09-144 | |||||||
| BRK(PTK6) | TK | Km bin. | 1mM | 08-165 | ||||||
| BRSK1 | STK | Km bin. | 1mM | Preincubation | 02-115 | |||||
| BRSK2 | STK | Km bin. | Preincubation | Cell Cycle | 02-116 | |||||
| BTK | TK | Km bin. | 1mM | 08-180 | ||||||
| BTK[C481S] | TK | Km bin. | 1mM | 08-547 | ||||||
| BUB1／BUB3 | STK | Km bin. | Preincubation | 05-187 | ||||||
| CaMK1α (CAMK1) | STK | Km bin. | 1mM | 02-104 | ||||||
| CaMK1δ (CAMK1D) | STK | Km bin. | 02-106 | |||||||
| CaMK2α(CAMK2A) | STK | Km bin. | Preincubation | 02-109 | ||||||
| CaMK2β(CAMK2B) | STK | Km bin. | Preincubation | 02-110 | ||||||
| CaMK2γ (CAMK2G) | STK | Km bin. | Preincubation | 02-112 | ||||||
| CaMK2δ (CAMK2D) | STK | Km bin. | Preincubation | 02-111 | ||||||
| CaMK4 | STK | Km bin. | 1mM | Preincubation | STK | 02-108 | ||||
| CDC2 /CycB1 | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 04-102 | ||||
| CDC7/ASK | STK | Km bin. | 1mM | Cell Cycle | 05-109 | |||||
| CDK2 /CycA2 | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 04-103 | |||
| CDK2 /CycE1 | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 04-165 | ||||
| CDK3 /CycE1 | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 04-104 | ||||
| CDK4／CycD3 | STK | Km bin. | 1mM | Cell Cycle | 04-105 | |||||
| CDK5／p25 | STK | Km bin. | 1mM | Preincubation | 04-106 | |||||
| CDK6／CycD3 | STK | Km bin. | 1mM | Cell Cycle | 04-107 | |||||
| CDK7／CycH／MAT1 | STK | Km bin. | 1mM | Cell Cycle | 04-108 | |||||
| CDK9／CycT1 | STK | Km bin. | 1mM | Cell Cycle | 04-110 | |||||
| CGK2 (PRKG2) | STK | Km bin. | Preincubation | 01-143 | ||||||
| CHK1(CHEK1) | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 02-117 | |||
| CHK2(CHEK2) | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 02-162 | ||||
| CK1α (CSNK1A1) | STK | Km bin. | 1mM | 03-101 | ||||||
| CK1γ1 (CSNK1G1) | STK | Km bin. | Preincubation | 03-105 | ||||||
| CK1γ2 (CSNK1G2) | STK | Km bin. | Preincubation | 03-106 | ||||||
| CK1γ3 (CSNK1G3) | STK | Km bin. | Preincubation | 03-107 | ||||||
| CK1δ (CSNK1D) | STK | Km bin. | Preincubation | 03-103 | ||||||
| CK1ε (CSNK1E) | STK | Km bin. | 1mM | STK | 03-104 | |||||
| CK2α1/β (CSNK2A1/B) | STK | Km bin. | 1mM | Preincubation | Cell Cycle | 05-184 | ||||
| CK2α2/β (CSNK2A2/B) | STK | Km bin. | Preincubation | Cell Cycle | 05-185 | |||||
| CLK1 | STK | Km bin. | 1mM | Preincubation | 04-126 | |||||
| CLK2 | STK | Km bin. | 1mM | Preincubation | 04-127 | |||||
| CLK3 | STK | Km bin. | Preincubation | 04-128 | ||||||
| COT (MAP3K8) | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-301 | ||||||
| CRIK (CIT) | STK | Km bin. | 01-104 | |||||||
| CSK | TK | Km bin. | 1mM | TK | 08-111 | |||||
| DAPK1 | STK | Km bin. | 1mM | Preincubation | STK | 02-134 | ||||
| DCAMKL2 | STK | Km bin. | 02-140 | |||||||
| DDR1 | TK | Km bin. | 1mM | 08-113 | ||||||
| DDR2 | TK | Km bin. | 1mM | 08-114 | ||||||
| DLK (MAP3K12) | STK |
1mM (Cascade) |
MAPK (Cascade) |
09-111 | ||||||
| DYRK1A | STK | Km bin. | 1mM | Preincubation | 04-130 | |||||
| DYRK1B | STK | Km bin. | 1mM | Preincubation | STK | 04-131 | ||||
| DYRK2 | STK | Km bin. | Preincubation | 04-132 | ||||||
| DYRK3 | STK | Km bin. | Preincubation | 04-133 | ||||||
| EEF2K | STK | Km bin. | 10-113 | |||||||
| EGFR | TK | Km bin. | 1mM | Preincubation | TK | 08-115 | ||||
EGFR[C797S／L858R]
|
TK | Km bin. | 1mM | 08-563 | ||||||
| EGFR[d746-750/T790M] | TK | Km bin. | 1mM | Preincubation | 08-528 | |||||
| EGFR[d746-750] | TK | Km bin. | 1mM | Preincubation | 08-527 | |||||
|
EGFR[d746-750／C797S]
|
TK | Km bin. | 1mM | Preincubation | 08-564 | |||||
|
EGFR[d746-750／T790M／C797S]
|
TK | 1mM | 08-565 | |||||||
| EGFR[D770_N771insNPG] | TK | Km bin. | 1mM | 08-553 | ||||||
| EGFR[L858R] | TK | Km bin. | 1mM | Preincubation | 08-502 | |||||
| EGFR[L861Q] | TK | Km bin. | 1mM | Preincubation | 08-513 | |||||
| EGFR[T790M] | TK | Km bin. | 1mM | Preincubation | 08-194 | |||||
|
EGFR[T790M／C797S／L858R]
|
TK | Km bin. | 1mM | 08-559 | ||||||
| EGFR[T790M／L858R] | TK | Km bin. | 1mM | Preincubation | 08-510 | |||||
| EML4-ALK | TK | Km bin. | 1mM | 08-516 | ||||||
| EPHA1 | TK | Km bin. | 1mM | Preincubation | 08-119 | |||||
| EPHA2 | TK | Km bin. | 1mM | Preincubation | TK | 08-121 | ||||
| EPHA3 | TK | Km bin. | 1mM | Preincubation | 08-122 | |||||
| EPHA4 | TK | Km bin. | 1mM | Preincubation | 08-123 | |||||
| EPHA5 | TK | Km bin. | 1mM | Preincubation | 08-124 | |||||
| EPHA6 | TK | Km bin. | 1mM | Preincubation | 08-125 | |||||
| EPHA7 | TK | Km bin. | 1mM | Preincubation | 08-126 | |||||
| EPHA8 | TK | Km bin. | 1mM | Preincubation | 08-127 | |||||
| EPHB1 | TK | Km bin. | 1mM | Preincubation | 08-128 | |||||
| EPHB2 | TK | Km bin. | 1mM | Preincubation | 08-129 | |||||
| EPHB3 | TK | Km bin. | 1mM | Preincubation | 08-130 | |||||
| EPHB4 | TK | Km bin. | 1mM | Preincubation | TK | 08-131 | ||||
| Erk1 (MAPK3) | STK | Km bin. | 1mM | Preincubation |
MAPK (Cascade) |
04-142 | ||||
| Erk2(MAPK1) | STK | Km bin. | 1mM | Preincubation | STK |
MAPK (Cascade) |
04-143 | |||
| Erk5(MAPK7) | STK | Km bin. | 1mM |
MAPK (Cascade) |
04-146 | |||||
| FAK (PTK2) | TK | Km bin. | 1mM | 08-137 | ||||||
| FER | TK | Km bin. | 1mM | Preincubation | 08-139 | |||||
| FES | TK | Km bin. | 1mM | Preincubation | 08-140 | |||||
| FGFR1 | TK | Km bin. | 1mM | Preincubation | TK | 08-133 | ||||
| FGFR1[V561M] | TK | Km bin. | 1mM | 08-536 | ||||||
| FGFR2 | TK | Km bin. | 1mM | Preincubation | 08-134 | |||||
| FGFR2[V564I] | TK | Km bin. | 1mM | Preincubation | 08-546 | |||||
| FGFR3 | TK | Km bin. | 1mM | 08-135 | ||||||
| FGFR3[K650E] | TK | Km bin. | 1mM | 08-501 | ||||||
| FGFR3[K650M] | TK | Km bin. | 1mM | 08-199 | ||||||
| FGFR3[V555L] | TK | Km bin. | 1mM | 08-548 | ||||||
| FGFR3[V555M] | TK | Km bin. | 1mM | 08-543 | ||||||
| FGFR4 | TK | Km bin. | 1mM | Preincubation | 08-136 | |||||
| FGFR4[N535K] | TK | Km bin. | 1mM | 08-524 | ||||||
| FGFR4[V550E] | TK | Km bin. | 1mM | 08-525 | ||||||
| FGFR4[V550L] | TK | Km bin. | 1mM | Preincubation | 08-526 | |||||
| FGR | TK | Km bin. | 1mM | Preincubation | 08-166 | |||||
| FLT1 | TK | Km bin. | 1mM | Preincubation | 08-189 | |||||
| FLT3 | TK | Km bin. | 1mM | TK | 08-154 | |||||
| FLT4 | TK | Km bin. | 1mM | Preincubation | 08-190 | |||||
| FMS (CSF1R) | TK | Km bin. | 1mM | 08-155 | ||||||
| FRK | TK | Km bin. | 1mM | Preincubation | 08-167 | |||||
| FYN [isoform a] | TK | Km bin. | 1mM | 08-168 | ||||||
| FYN [isoform b] | TK | Km bin. | 1mM | 08-531 | ||||||
| GSK3α (GSK3A) | STK | Km bin. | 1mM | Preincubation | 04-140 | |||||
| GSK3β(GSK3B) | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 04-141 | |||
| Haspin (GSG2) | STK | Km bin. | Preincubation | 05-111 | ||||||
| HCK | TK | Km bin. | 1mM | 08-169 | ||||||
| HER2 | TK | Km bin. | 1mM | 08-016 | ||||||
| HER4 (ERBB4) | TK | Km bin. | 1mM | Preincubation | 08-118 | |||||
| HGK (MAP4K4) | STK | Km bin. | 1mM | STK | 07-137 | |||||
| HIPK1 | STK | Km bin. | Preincubation | 04-135 | ||||||
| HIPK2 | STK | Km bin. | Preincubation | 04-136 | ||||||
| HIPK3 | STK | Km bin. | Preincubation | 04-137 | ||||||
| HIPK4 | STK | Km bin. | 1mM | Preincubation | 04-138 | |||||
|
HPK1(MAP4K1)
|
STK | Km bin. | 07-410 | |||||||
| IGF1R | TK | Km bin. | 1mM | Preincubation | TK | 08-141 | ||||
| IKKα(CHUK) | STK | Km bin. | 05-112 | |||||||
| IKKβ (IKBKB) | STK | Km bin. | 1mM | Preincubation | STK | 05-084 | ||||
| IKKε (IKBKE) | STK | Km bin. | 05-114 | |||||||
| INSR | TK | Km bin. | 1mM | Preincubation | 08-142 | |||||
| IRAK1 | STK | Km bin. | 09-101 | |||||||
| IRAK4 | STK | Km bin. | 1mM | STK | 09-145 | |||||
| IRR (INSRR) | TK | Km bin. | 1mM | 08-143 | ||||||
| ITK | TK | Km bin. | 1mM | TK | 08-181 | |||||
| JAK1 | TK | Km bin. | 1mM | 08-144 | ||||||
| JAK2 | TK | Km bin. | 1mM | Preincubation | 08-045 | |||||
| JAK3 | TK | Km bin. | 1mM | Preincubation | TK | 08-046 | ||||
| JNK1(MAPK8) | STK | Km bin. | 1mM | Preincubation |
MAPK (Cascade) |
04-163 | ||||
| JNK2(MAPK9) | STK | Km bin. | 1mM | Preincubation | STK |
MAPK (Cascade) |
04-164 | |||
| JNK3 (MAPK10) | STK | Km bin. | 1mM | Preincubation |
MAPK (Cascade) |
04-150 | ||||
| KDR | TK | Km bin. | 1mM | Preincubation | TK | 08-191 | ||||
| KIT | TK | Km bin. | 1mM | 08-156 | ||||||
| KIT[D816E] | TK | Km bin. | 1mM | 08-541 | ||||||
| KIT[D816V] | TK | Km bin. | 1mM | 08-505 | ||||||
| KIT[D816Y] | TK | Km bin. | 1mM | 08-534 | ||||||
| KIT[T670I] | TK | Km bin. | 1mM | 08-195 | ||||||
| KIT[V560G] | TK | Km bin. | 1mM | 08-504 | ||||||
| KIT[V654A] | TK | Km bin. | 1mM | 08-511 | ||||||
| LATS2 | STK | Km bin. | 01-124 | |||||||
| LCK | TK | Km bin. | 1mM | Preincubation | TK | 08-170 | ||||
| LOK (STK10) | STK | Km bin. | 07-315 | |||||||
| LTK | TK | Km bin. | 1mM | 08-106 | ||||||
| LYNa | TK | Km bin. | 1mM | Preincubation | 08-171 | |||||
| LYNb | TK | Km bin. | 1mM | Preincubation | 08-172 | |||||
| MAP2K1 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-141 | ||||||
| MAP2K2 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-142 | ||||||
| MAP2K3 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-143 | ||||||
| MAP2K4 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-144 | ||||||
| MAP2K5 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-145 | ||||||
| MAP2K6 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-146 | ||||||
| MAP2K7 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-148 | ||||||
| MAP3K1 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-103 | ||||||
| MAP3K2 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-104 | ||||||
| MAP3K3 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-105 | ||||||
| MAP3K4 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-106 | ||||||
| MAP3K5 | STK |
1mM (Cascade) |
MAPK (Cascade) |
07-107 | ||||||
| MAP4K2 | STK | Km bin. | 07-111 | |||||||
| MAPKAPK2 | STK | Km bin. | 1mM | Preincubation | STK | 02-142 | ||||
| MAPKAPK3 | STK | Km bin. | Preincubation | 02-143 | ||||||
| MAPKAPK5 | STK | Km bin. | Preincubation | 02-144 | ||||||
| MARK1 | STK | Km bin. | Preincubation | 02-120 | ||||||
| MARK2 | STK | Km bin. | Preincubation | 02-121 | ||||||
| MARK3 | STK | Km bin. | Preincubation | 02-122 | ||||||
| MARK4 | STK | Km bin. | Preincubation | 02-123 | ||||||
| MELK | STK | Km bin. | 02-124 | |||||||
| MER (MERTK) | TK | Km bin. | 1mM | Preincubation | 08-108 | |||||
| MET | TK | Km bin. | 1mM | Preincubation | TK | 08-151 | ||||
| MET[D1228H] | TK | Km bin. | 1mM | Preincubation | 08-540 | |||||
| MET[M1250T] | TK | Km bin. | 1mM | Preincubation | 08-545 | |||||
| MET[Y1235D] | TK | Km bin. | 1mM | Preincubation | 08-198 | |||||
| MINK (MINK1) | STK | Km bin. | 1mM | 07-139 | ||||||
| MLK1(MAP3K9) | STK |
1mM (Cascade) |
MAPK (Cascade) |
09-115 | ||||||
| MLK2(MAP3K10) | STK |
1mM (Cascade) |
MAPK (Cascade) |
09-116 | ||||||
| MLK3(MAP3K11) | STK |
1mM (Cascade) |
MAPK (Cascade) |
09-017 | ||||||
| MNK1 (MKNK1) | STK | Km bin. | Preincubation | 02-145 | ||||||
| MNK2 (MKNK2) | STK | Km bin. | Preincubation | 02-146 | ||||||
| MOS | STK |
1mM (Cascade) |
MAPK (Cascade) |
05-118 | ||||||
| MRCKα (CDC42BPA) | STK | Km bin. | 01-107 | |||||||
| MRCKβ (CDC42BPB) | STK | Km bin. | 01-108 | |||||||
| MSK1 (RPS6KA5) | STK | Km bin. | Preincubation | 01-147 | ||||||
| MSK2 (RPS6KA4) | STK | Km bin. | 01-148 | |||||||
| MSSK1 (STK23) | STK | Km bin. | 04-159 | |||||||
| MST1 (STK4) | STK | Km bin. | 1mM | STK | 07-116 | |||||
| MST2 (STK3) | STK | Km bin. | 07-117 | |||||||
| MST3 (STK24) | STK | Km bin. | 07-118 | |||||||
| MST4 | STK | Km bin. | 07-119 | |||||||
| MUSK | TK | Km bin. | 1mM | 08-153 | ||||||
| NDR1 (STK38) | STK | Km bin. | 01-125 | |||||||
| NDR2 (STK38L) | STK | Km bin. | 01-126 | |||||||
| NEK1 | STK | Km bin. | 1mM | Cell Cycle | 05-123 | |||||
| NEK2 | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 05-226 | |||
| NEK4 | STK | Km bin. | Preincubation | 05-128 | ||||||
| NEK6 | STK | Km bin. | 1mM | Cell Cycle | 05-130 | |||||
| NEK7 | STK | Km bin. | 1mM | Cell Cycle | 05-131 | |||||
| NEK9 | STK | Km bin. | 1mM | Cell Cycle | 05-133 | |||||
| NIM1K(MGC42105) | STK | Km bin. | Preincubation | 02-175 | ||||||
| NPM1-ALK | TK | Km bin. | 1mM | Preincubation | 08-517 | |||||
| NuaK1 | STK | Km bin. | Preincubation | 02-126 | ||||||
| NuaK2 | STK | Km bin. | Preincubation | 02-127 | ||||||
| p38α(MAPK14) | STK | Km bin. | 1mM | Preincubation | STK |
MAPK (Cascade) |
Cell Cycle | 04-152 | ||
| p38β (MAPK11) | STK | Km bin. | 1mM | Preincubation |
MAPK (Cascade) |
04-153 | ||||
| p38γ (MAPK12) | STK | Km bin. | 1mM | Preincubation |
MAPK (Cascade) |
04-155 | ||||
| p38δ (MAPK13) | STK | Km bin. | 1mM | Preincubation |
MAPK (Cascade) |
04-154 | ||||
| p70S6K(RPS6KB1) | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 01-154 | |||
| p70S6Kβ(RPS6KB2) | STK | Km bin. | Preincubation | 01-155 | ||||||
| PAK1 | STK | Km bin. | Preincubation | 07-123 | ||||||
| PAK2 | STK | Km bin. | 1mM | Preincubation | STK | 07-124 | ||||
| PAK4 | STK | Km bin. | 07-126 | |||||||
| PAK5 (PAK7) | STK | Km bin. | Preincubation | 07-127 | ||||||
| PAK6 | STK | Km bin. | 07-128 | |||||||
| PASK | STK | Km bin. | 02-128 | |||||||
| PBK | STK | Km bin. | 1mM | STK | 05-168 | |||||
| PDGFRα(PDGFRA) | TK | Km bin. | 1mM | Preincubation | TK | 08-157 | ||||
| PDGFRα(PDGFRA)[D842V] | TK | Km bin. | 1mM | Preincubation | 08-506 | |||||
| PDGFRα(PDGFRA)[T674I] | TK | Km bin. | 1mM | 08-503 | ||||||
| PDGFRα(PDGFRA)[V561D] | TK | Km bin. | 1mM | Preincubation | 08-507 | |||||
| PDGFRβ (PDGFRB) | TK | Km bin. | 1mM | Preincubation | 08-158 | |||||
| PDHK2 (PDK2) | STK | Km bin. | 10-140 | |||||||
| PDHK4 (PDK4) | STK | Km bin. | 10-125 | |||||||
| PDK1(PDPK1) | STK | Km bin. | 1mM | STK | 01-132 | |||||
| PEK (EIF2AK3) | STK | Km bin. | 05-155 | |||||||
| PGK (PRKG1) | STK | Km bin. | 01-142 | |||||||
| PHKG1 | STK | Km bin. | 02-152 | |||||||
| PHKG2 | STK | Km bin. | 02-153 | |||||||
| PIM1 | STK | Km bin. | 1mM | Preincubation | STK | Cell Cycle | 02-054 | |||
| PIM2 | STK | Km bin. | 1mM | Cell Cycle | 02-155 | |||||
| PIM3 | STK | Km bin. | 02-156 | |||||||
| PKACα(PRKACA) | STK | Km bin. | 1mM | STK | 01-127 | |||||
| PKACβ (PRKACB) | STK | Km bin. | 01-128 | |||||||
| PKACγ (PRKACG) | STK | Km bin. | 01-129 | |||||||
| PKCα(PRKCA) | STK | Km bin. | 1mM | STK | 01-133 | |||||
| PKCβ1(PRKCB1) | STK | Km bin. | 01-134 | |||||||
| PKCβ2(PRKCB2) | STK | Km bin. | 01-165 | |||||||
| PKCγ(PRKCG) | STK | Km bin. | 01-137 | |||||||
| PKCδ(PRKCD) | STK | Km bin. | Preincubation | 01-135 | ||||||
| PKCε(PRKCE) | STK | Km bin. | 1mM | Preincubation | 01-136 | |||||
| PKCζ (PRKCZ) | STK | Km bin. | Preincubation | 01-141 | ||||||
| PKCη (PRKCH) | STK | Km bin. | Preincubation | 01-138 | ||||||
| PKCθ(PRKCQ) | STK | Km bin. | 01-140 | |||||||
| PKCι (PRKCI) | STK | Km bin. | 01-139 | |||||||
| PKD1 (PRKD1) | STK | Km bin. | Preincubation | 02-157 | ||||||
| PKD2 (PRKD2) | STK | Km bin. | 1mM | Preincubation | STK | 02-158 | ||||
| PKD3 (PRKD3) | STK | Km bin. | 02-159 | |||||||
| PKN1 | STK | Km bin. | 01-144 | |||||||
| PKR (EIF2AK2) | STK | Km bin. | 05-156 | |||||||
| PLK1 | STK | Km bin. | 1mM | Cell Cycle | 05-157 | |||||
| PLK2 | STK | Km bin. | Cell Cycle | 05-158 | ||||||
| PLK3 | STK | Km bin. | 1mM | 05-159 | ||||||
| PRKX | STK | Km bin. | 01-130 | |||||||
| PYK2 (PTK2B) | TK | Km bin. | 1mM | Preincubation | TK | 08-138 | ||||
| QIK (SNF1LK2) | STK | Km bin. | 1mM | Preincubation | 02-129 | |||||
| RAF1 | STK |
1mM (Cascade) |
MAPK (Cascade) |
09-125 | ||||||
| RET | TK | Km bin. | 1mM | Preincubation | 08-159 | |||||
| RET[G691S] | TK | Km bin. | 1mM | Preincubation | 08-522 | |||||
| RET[M918T] | TK | Km bin. | 1mM | Preincubation | 08-508 | |||||
| RET[S891A] | TK | Km bin. | 1mM | Preincubation | 08-523 | |||||
| RET[Y791F] | TK | Km bin. | 1mM | Preincubation | 08-521 | |||||
| ROCK1 | STK | Km bin. | 1mM | STK | 01-109 | |||||
| ROCK2 | STK | Km bin. | Preincubation | 01-110 | ||||||
| RON (MST1R) | TK | Km bin. | 1mM | Preincubation | 08-152 | |||||
| ROS (ROS1) | TK | Km bin. | 1mM | Preincubation | 08-163 | |||||
| RSK1 (RPS6KA1) | STK | Km bin. | 1mM | Cell Cycle | 01-149 | |||||
| RSK2(RPS6KA3) | STK | Km bin. | Preincubation | 01-150 | ||||||
| RSK3 (RPS6KA2) | STK | Km bin. | 1mM | Preincubation | 01-151 | |||||
| RSK4 (RPS6KA6) | STK | Km bin. | 1mM | Preincubation | 01-152 | |||||
| SGK | STK | Km bin. | 1mM | Preincubation | STK | 01-158 | ||||
| SGK2 | STK | Km bin. | 01-159 | |||||||
| SGK3 (SGKL) | STK | Km bin. | Preincubation | 01-160 | ||||||
| SIK (SNF1LK) | STK | Km bin. | 1mM | 02-131 | ||||||
| skMLCK (MYLK2) | STK | Km bin. | 1mM | Preincubation | 02-150 | |||||
| SLK | STK | Km bin. | 07-129 | |||||||
| SPHK1 | Lipid | Km bin. | Preincubation | 11-105 | ||||||
| SPHK2 | Lipid | Km bin. | 11-106 | |||||||
| SRC | TK | Km bin. | 1mM | Preincubation | TK | 08-173 | ||||
| SRM (SRMS) | TK | Km bin. | 1mM | Preincubation | 08-174 | |||||
| SRPK1 | STK | Km bin. | 04-160 | |||||||
| SRPK2 | STK | Km bin. | 04-161 | |||||||
| SYK | TK | Km bin. | 1mM | TK | 08-176 | |||||
| TAK1-TAB1(MAP3K7) | STK |
1mM (Cascade) |
MAPK (Cascade) |
09-019 | ||||||
| TAOK2 | STK | Km bin. | 07-133 | |||||||
| TBK1 | STK | Km bin. | Preincubation | 05-115 | ||||||
| TEC | TK | Km bin. | 1mM | Preincubation | 08-182 | |||||
| TIE2 (TEK) | TK | Km bin. | 1mM | Preincubation | TK | 08-185 | ||||
| TNIK | STK | Km bin. | 1mM | 07-138 | ||||||
| TNK1 | TK | Km bin. | 1mM | 08-104 | ||||||
| TRKA (NTRK1) | TK | Km bin. | 1mM | TK | 08-186 | |||||
| TRKB(NTRK2) | TK | Km bin. | 1mM | Preincubation | 08-187 | |||||
| TRKC (NTRK3) | TK | Km bin. | 1mM | Preincubation | 08-197 | |||||
| TSSK1 | STK | Km bin. | 1mM | Preincubation | STK | 02-364 | ||||
| TSSK2 | STK | Km bin. | 02-165 | |||||||
| TSSK3 | STK | Km bin. | 02-166 | |||||||
| TXK | TK | Km bin. | 1mM | 08-183 | ||||||
| TYK2 | TK | Km bin. | 1mM | 08-147 | ||||||
| TYRO3 | TK | Km bin. | 1mM | Preincubation | TK | 08-109 | ||||
| WNK1 | STK | Km bin. | 05-179 | |||||||
| WNK2 | STK | Km bin. | 05-180 | |||||||
| WNK3 | STK | Km bin. | 05-181 | |||||||
| YES(YES1) | TK | Km bin. | 1mM | Preincubation | 08-175 | |||||
| YES(YES1)[T348I] | TK | Km bin. | 1mM | Preincubation | 08-533 | |||||
| ZAP70 | TK | Km bin. | 1mM | 08-177 | ||||||
